Advancing the antituberculosis activity of nitropicolinic acids and amides

WHO

World Health Organisation

DprE1

decaprenylphosphoryl-β-d-ribose 2′-oxidase

DprE2

decaprenylphosphoryl-2-keto-β-d-erythropentose reductase

M. tb

Mycobacterium tuberculosis

Ddn

deazaflavin-dependent nitroreductase

HATU

hexafluorophosphate azabenzotriazole tetramethyl uronium

DIPEA

N,N-diisopropylethylamine

CC50

half-maximum cytotoxic concentration

FIC

fractional inhibitory concentration

LipE

lipophilic efficiency

LORA

low-oxygen-recovery assay

MABA

microplate alamar blue assay

MBC

minimum bactericidal concentration

PAE

post-antibiotic effect

TMM

trehalose monomycolates

PE

phosphatidylethanolamine

PIMs

phosphatidylinositol mannosides

FAME

fatty acid methyl esters

MAME

mycolic acid methyl esters

APCI

atmospheric pressure chemical ionisation

Comments (0)

No login
gif