Evaluation of Newly Synthesized Compounds Targeting Carbonic Anhydrase Enzyme for Antineoplastic Activity in Solid Tumors

Bukowski, K., M. Kciuk, and R. Kontek, Mechanisms of multidrug resistance in cancer chemotherapy. International journal of molecular sciences, 2020. 21(9): p. 3233.

Sunjuk, M., et al., Transition Metal Complexes of Schiff Base Ligands Prepared from Reaction of Aminobenzothiazole with Benzaldehydes. Inorganics, 2022. 10(4): p. 43.

Mansoori, B., et al., The different mechanisms of cancer drug resistance: a brief review. Advanced pharmaceutical bulletin, 2017. 7(3): p. 339.

Dallavalle, S., et al., Improvement of conventional anti-cancer drugs as new tools against multidrug resistant tumors. Drug Resistance Updates, 2020. 50: p. 100682.

Butturini, E., et al., Tumor dormancy and interplay with hypoxic tumor microenvironment. International journal of molecular sciences, 2019. 20(17): p. 4305.

Mussi, S., et al., Antiproliferative effects of sulphonamide carbonic anhydrase inhibitors C18, SLC-0111 and acetazolamide on bladder, glioblastoma and pancreatic cancer cell lines. Journal of Enzyme Inhibition and Medicinal Chemistry, 2022. 37(1): p. 280-286.

Supuran, C.T., Structure and function of carbonic anhydrases. Biochemical Journal, 2016. 473(14): p. 2023-2032.

Angeli, A., et al., Pyrazolo [4, 3-c] pyridine Sulfonamides as Carbonic Anhydrase Inhibitors: Synthesis, Biological and In Silico Studies. Pharmaceuticals, 2022. 15(3): p. 316.

Khushal, A., et al., Synthesis, carbonic anhydrase II/IX/XII inhibition, DFT, and molecular docking studies of hydrazide-sulfonamide hybrids of 4-methylsalicyl-and acyl-substituted hydrazide. BioMed Research International, 2022. 2022.

Supuran, C.T., et al., Carbonic anhydrase inhibitors: sulfonamides as antitumor agents? Bioorganic & medicinal chemistry, 2001. 9(3): p. 703-714.

Supuran, C.T., Experimental carbonic anhydrase inhibitors for the treatment of hypoxic tumors. Journal of Experimental Pharmacology, 2020: p. 603-617.

Angeli, A., et al., Carbonic anhydrase inhibitors targeting metabolism and tumor microenvironment. Metabolites, 2020. 10(10): p. 412.

Said, M.A., et al., Sulfonamide-based ring-fused analogues for CAN508 as novel carbonic anhydrase inhibitors endowed with antitumor activity: Design, synthesis, and in vitro biological evaluation. European Journal of Medicinal Chemistry, 2020. 189: p. 112019.

Borcea, A.-M., et al., An overview of the synthesis and antimicrobial, antiprotozoal, and antitumor activity of thiazole and bisthiazole derivatives. Molecules, 2021. 26(3): p. 624.

Sharma, P.C., et al., Thiazole-containing compounds as therapeutic targets for cancer therapy. European journal of medicinal chemistry, 2020. 188: p. 112016.

Ramos-Inza, S., et al., Thiazole moiety: An interesting scaffold for developing new antitumoral compounds, in Heterocycles-synthesis and biological activities. 2019, IntechOpen.

Arshad, M.F., et al., Thiazole: A versatile standalone moiety contributing to the development of various drugs and biologically active agents. Molecules, 2022. 27(13): p. 3994.

Supuran, C.T., A. Scozzafava, and A. Casini, Carbonic anhydrase inhibitors. Medicinal research reviews, 2003. 23(2): p. 146-189.

Billah, M.M., et al., Determination of the presence and pharmacokinetic profile of ciprofloxacin by TLC and HPLC method respectively in broiler chicken after single oral administration. The Journal of Antibiotics, 2014. 67(11): p. 745-748.

Saeedi, M., et al., Synthesis and biological investigation of some novel sulfonamide and amide derivatives containing coumarin moieties. Iranian Journal of Pharmaceutical Research: IJPR, 2014. 13(3): p. 881.

Jawad, H.A., et al., Design, Synthesis, In Silico Study And Preliminary Pharmacological Assessment Of New Ciprofloxacin Analogues Having Thiazole Nucleus. Journal of Pharmaceutical Negative Results, 2023: p. 91-104.

Park, H.-S., et al., Synthesis and characterization of novel hydantoins as potential COX-2 inhibitors: 1, 5-Diarylhydantoins. Bulletin of the Korean Chemical Society, 2007. 28(5): p. 751-757.

留言 (0)

沒有登入
gif